翻訳と辞書
Words near each other
・ A-normal form
・ A-not-A question
・ A-not-B error
・ A-ok
・ A-One (band)
・ A-One (TV channel)
・ A-366,833
・ A-372159
・ A-40174
・ A-412,997
・ A-41988
・ A-423,579
・ A-68930
・ A-7 & A-10 (Arizona)
・ A-77636
A-796,260
・ A-834,735
・ A-836,339
・ A-84,543
・ A-86929
・ A-90 Orlyonok
・ A-91
・ A-971432
・ A-A line
・ A-A-P
・ A-Acayipsin
・ A-B Emblem
・ A-B Helicopters A/W 95
・ A-b-c-darian
・ A-Ba-Ni-Bi


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A-796,260 : ウィキペディア英語版
A-796,260

A-796,260 is a drug developed by Abbott Laboratories that acts as a potent and selective cannabinoid CB2 receptor agonist. Replacing the aromatic 3-benzoyl or 3-naphthoyl group found in most indole derived cannabinoids with the 3-tetramethylcyclopropylmethanone group, imparts significant selectivity for CB2, and A-796,260 was found to be a highly selective CB2 agonist with little affinity for CB1, having a CB2 Ki of 4.6 nM vs 945 nM at CB1.〔
〕 It has potent analgesic and anti-inflammatory actions in animal models, being especially effective in models of neuropathic pain, but without producing cannabis-like behavioral effects.
==Legal Status==

As of October 2015 A-796,260 is a controlled substance in China.

抄文引用元・出典: フリー百科事典『 ウィキペディア(Wikipedia)
ウィキペディアで「A-796,260」の詳細全文を読む



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