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AM-1248
AM-1248 is a drug that acts as a moderately potent agonist for both the cannabinoid receptors CB1 and CB2, but with some dispute between sources over its exact potency and selectivity. Replacing the 3-(1-naphthoyl) group found in many indole derived cannabinoid ligands, with an adamantoyl group, generally confers significant CB2 selectivity,〔 〕 but reasonable CB1 affinity and selectivity is retained when an N-methylpiperidin-2-ylmethyl substitution is used at the indole 1-position. The related compound 1-pentyl-3-(1-adamantoyl)indole was identified as having been sold as a cannabinoid designer drug in Hungary in 2011, along with another synthetic cannabinoid AM-679. ==Legality== Sweden's public health agency suggested to classify AM-1248 as hazardous substance on June 1, 2015.〔(【引用サイトリンク】 title=23 nya ämnen kan klassas som narkotika eller hälsofarlig vara )〕 As of October 2015 AM-1248 is a controlled substance in China.
抄文引用元・出典: フリー百科事典『 ウィキペディア(Wikipedia)』 ■ウィキペディアで「AM-1248」の詳細全文を読む
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