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AM-906
AM-906 is an analgesic drug which is a cannabinoid agonist with a conformationally restricted side chain. It is a potent and selective agonist for the CB1 cannabinoid receptor, with a Ki of 0.8nM at CB1 and 9.5nM at CB2, a selectivity of almost 12x.〔Papahatjis DP, ''et al.'' Pharmacophoric requirements for cannabinoid side chains: multiple bond and C1'-substituted delta 8-tetrahydrocannabinols. ''Journal of Medicinal Chemistry''. 1998 Mar 26;41(7):1195-200. PMID 9544219〕 ==See also==
* AM-1235 * AM-2389
抄文引用元・出典: フリー百科事典『 ウィキペディア(Wikipedia)』 ■ウィキペディアで「AM-906」の詳細全文を読む
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