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BD1018
BD1018 or (S)-2-()octahydropyrrolo()pyrazine is a selective sigma receptor ligand, with a reported binding affinity of ''K''i = 5 ± 0.7 nM for the sigma-1 receptor and approximately 10 times selectivity over the sigma-2 receptor. Unlike its enantiomer, BD1031, BD1018 acts as a sigma receptor antagonist.〔 Consistent with other reported sigma receptor antagonists, BD1018 deccreases the behavioural toxicity of cocaine in Swiss Webster mice.〔 ==See also==
* BD1008 * BD1031
抄文引用元・出典: フリー百科事典『 ウィキペディア(Wikipedia)』 ■ウィキペディアで「BD1018」の詳細全文を読む
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