翻訳と辞書
Words near each other
・ Cid
・ CID (Indian TV series)
・ CID 72
・ Cid Corman
・ Cid Edwards
・ Cid Formation
・ Cid Gomes
・ Cid Moreira
・ Cid Nascimento
・ Cid Ricketts Sumner
・ Cid Samson
・ CID Shankar
・ CID The Dummy
・ CID Unnikrishnan B.A., B.Ed.
・ Cid, North Carolina
CID-16020046
・ CID-42
・ CID-85469571
・ CIDA
・ CIDA City Campus
・ CIDAC
・ Cidacos
・ Cidade Ademar
・ Cidade Ademar (district of São Paulo)
・ Cidade Ameaçada
・ Cidade Baixa (disambiguation)
・ Cidade Baixa, Porto Alegre
・ Cidade da Maia
・ Cidade das Artes
・ Cidade de Deus (Osasco)


Dictionary Lists
翻訳と辞書 辞書検索 [ 開発暫定版 ]
スポンサード リンク

CID-16020046 : ウィキペディア英語版
CID-16020046

CID-16020046 is a compound which acts as an inverse agonist at the former orphan receptor GPR55, and may be the first selective inverse agonist characterised for this receptor. It was found to block a number of GPR55 mediated responses such as wound healing and activation of immune system T-cells and B-cells, as well as showing inverse agonist activity in the absence of GPR55 agonist stimulation. However while it was found to have good selectivity over the related CB1 and CB2 cannabinoid receptors as well as a number of other targets, CID-16020046 has not yet been tested against another related receptor GPR18, so its selectivity for GPR55 over this target has not been established.〔Kargl J, Brown AJ, Andersen L, Dorn G, Schicho R, Waldhoer M, Heinemann A. A selective antagonist reveals a potential role of G protein-coupled receptor 55 in platelet and endothelial cell function. ''Journal of Pharmacology and Experimental Therapeutics''. 2013 Jul;346(1):54-66. DOI 10.1124/jpet.113.204180. PMID 23639801〕
==See also==

* CID-85469571
* O-1918
* PSB-SB-487

抄文引用元・出典: フリー百科事典『 ウィキペディア(Wikipedia)
ウィキペディアで「CID-16020046」の詳細全文を読む



スポンサード リンク
翻訳と辞書 : 翻訳のためのインターネットリソース

Copyright(C) kotoba.ne.jp 1997-2016. All Rights Reserved.