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翻訳と辞書　辞書検索 [ 開発暫定版 ] スポンサード リンク Cyprodime ： ウィキペディア英語版 Cyprodime Cyprodime is an opioid antagonist from the morphinan family of drugs. Cyprodime is a selective opioid antagonist which blocks the μ-opioid receptor,〔Schmidhammer H, Burkard WP, Eggstein-Aeppli L, Smith CF. Synthesis and biological evaluation of 14-alkoxymorphinans. 2. (−)-N- (cyclopropylmethyl)- 4,14-dimethoxymorphinan- 6-one, a selective mu opioid receptor antagonist. ''Journal of Medicinal Chemistry''. 1989 Feb;32(2):418-21. PMID 2536439〕 but without affecting the δ-opioid or κ-opioid receptors. This makes it useful for scientific research as it allows the μ-opioid receptor to be selectively deactivated so that the actions of the δ and κ receptors can be studied separately, in contrast to better known opioid antagonists such as naloxone which block all three opioid receptor subtypes.〔Márki A, Monory K, Otvös F, Tóth G, Krassnig R, Schmidhammer H, Traynor JR, Roques BP, Maldonado R, Borsodi A. Mu-opioid receptor specific antagonist cyprodime: characterization by in vitro radioligand and ()GTPgammaS binding assays. ''European Journal of Pharmacology''. 1999 Oct 27;383(2):209-14. PMID 10585536〕 ==See also== * Samidorphan 抄文引用元・出典: フリー百科事典『 ウィキペディア（Wikipedia）』 ■ウィキペディアで「Cyprodime」の詳細全文を読む スポンサード リンク 翻訳と辞書 : 翻訳のためのインターネットリソース Copyright(C) kotoba.ne.jp 1997-2016. All Rights Reserved.