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Fluorophen
Fluorophen (fluorofen) is a fluorinated analog of phenazocine, an opioid drug of the benzomorphan family, which was developed as a radioligand for the purpose of labeling opioid receptors during PET scans (with 18F). Unlike most other benzomorphan derivatives, fluorophen acts as a full agonist of the opioid receptors with preferential affinity for the μ-opioid receptor (approximately 6x that of morphine), similar but slightly lower affinity for the δ-opioid receptor (equipotent to (D-Leu5 )enkephalin), and very low affinity for the κ-opioid receptor.〔〔 == See also ==
* Benzomorphan
抄文引用元・出典: フリー百科事典『 ウィキペディア(Wikipedia)』 ■ウィキペディアで「Fluorophen」の詳細全文を読む
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