翻訳と辞書 Words near each other ・ Gabarret ・ Gabarus ・ Gabarus Lake ・ Gabarus Lake, Nova Scotia ・ Gabas ・ Gabas (river) ・ Gabas, Pyrénées-Atlantiques ・ Gabasawa ・ Gabasheane Masupha ・ Gabashvili ・ Gabaston ・ Gabat ・ Gabata ・ Gabay ・ Gabazeleh ・ Gabazine ・ Gabb ・ Gabb's snail ・ Gabba ・ Gabba (band) ・ Gabba Front Berlin ・ Gabba Gabba Hey ・ Gabba Island (Queensland) ・ Gabbai ・ Gabbala ・ Gabbang ・ Gabbar Is Back ・ Gabbar Singh ・ Gabbar Singh (character) ・ Gabbar Singh (field hockey) Dictionary Lists mini英和辞書 mini和英辞書 Webster 1913 Latin-English FOLDOC Wikipedia English ウィキペディア

翻訳と辞書　辞書検索 [ 開発暫定版 ] スポンサード リンク Gabazine ： ウィキペディア英語版 Gabazine Gabazine (SR-95531) is a drug that acts as an antagonist at GABAA receptors. It is used in scientific research and has no role in medicine, as it would be expected to produce convulsions if used in humans. Gabazine binds to the GABA recognition site of the receptor-channel complex and acts as an allosteric inhibitor of channel opening. The net effect is to reduce GABA-mediated synaptic inhibition by inhibiting chloride flux across the cell membrane, and thus inhibiting neuronal hyperpolarization. While phasic (synaptic) inhibition is gabazine-sensitive, tonic (extrasynaptic) inhibition is relatively gabazine-insensitive. Gabazine has been found to bind to and antagonize α4βδ subunit-containing GABAA receptors, which may represent the GHB receptor. ==References== 抄文引用元・出典: フリー百科事典『 ウィキペディア（Wikipedia）』 ■ウィキペディアで「Gabazine」の詳細全文を読む スポンサード リンク 翻訳と辞書 : 翻訳のためのインターネットリソース Copyright(C) kotoba.ne.jp 1997-2016. All Rights Reserved.