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JWH-210
JWH-210 is an analgesic chemical from the naphthoylindole family, which acts as a potent cannabinoid agonist at both the CB1 and CB2 receptors, with Ki values of 0.46nM at CB1 and 0.69nM at CB2. It is one of the most potent 4-substituted naphthoyl derivatives in the naphthoylindole series, having a higher binding affinity (i.e. lower Ki) at CB1 than both its 4-methyl and 4-''n''-propyl homologues JWH-122 (CB1 Ki 0.69nM) and JWH-182 (CB1 Ki 0.65nM) respectively, and than the 4-methoxy compound JWH-081 (CB1 Ki 1.2nM).〔
〕 It was discovered by and named after Dr. John W. Huffman.
==Legal Status==
JWH-210 and JWH-122 were banned in Sweden on 1 October 2010 as hazardous goods harmful to health, after being identified as ingredients in "herbal" synthetic cannabis products.〔(Swedish Code of Statutes Regulation (2010:1086). )〕〔(Swedish Code of Statutes Regulation (2010:1086). (pdf) )〕 The substances JWH-210, JWH-122 and JWH-203 were classified as illegal drugs by the Swedish government as of 1 September 2011.〔LVFS 2011:8〕
As of October 2015 JWH-210 is a controlled substance in China.
抄文引用元・出典: フリー百科事典『 ウィキペディア（Wikipedia）』
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