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|Section2= |Section3= }} VUF-5681 is a potent and selective histamine antagonist which binds selectively to the H3 subtype.〔Moreno-Delgado D, Torrent A, Gómez-Ramírez J, de Esch I, Blanco I, Ortiz J. Constitutive activity of H3 autoreceptors modulates histamine synthesis in rat brain through the cAMP/PKA pathway. ''Neuropharmacology''. 2006 Sep;51(3):517-23. PMID 16769092〕 However while VUF-5681 blocks the activity of more potent H3 agonists, recent studies suggest that it may have some weak partial agonist activity when administered by itself. ==References== 〔 抄文引用元・出典: フリー百科事典『 ウィキペディア(Wikipedia)』 ■ウィキペディアで「VUF-5681」の詳細全文を読む スポンサード リンク
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