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Fludiazepam, marketed under the brand name Erispan〔(【引用サイトリンク】 title=Benzodiazepine Names )〕 is a potent benzodiazepine and 2'-fluoro derivative of diazepam, originally developed by Hoffman-La Roche in the 1960s.〔US Patent 3299053 -ARYL-JH-L,X-BENZODIAZEPIN-Z(LH)-ONES〕 It is marketed in Japan and Taiwan in the form of 0.25 mg tablets, making it around 40x more potent than diazepam. It exerts its pharmacological properties via enhancement of GABAergic inhibition. Fludiazepam has 4 times more binding affinity for benzodiazepine receptors than diazepam. It possesses anxiolytic, anticonvulsant, sedative, hypnotic and skeletal muscle relaxant properties. As with all benzodiazepines, fludiazepam is used recreationally. ==See also== *Benzodiazepine *Diazepam *Diclazepam (the 2'-chloro-analogue). *Flunitrazepam (the 7-nitro-analogue). 抄文引用元・出典: フリー百科事典『 ウィキペディア（Wikipedia）』 ■ウィキペディアで「fludiazepam」の詳細全文を読む スポンサード リンク
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