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phenomorphan
Phenomorphan is an opioid analgesic. It is not currently used in medicine, but has similar side-effects to other opiates, which include itching, nausea and respiratory depression.
Phenomorphan is a highly potent drug due to the N-phenethyl group, which boosts affinity to the μ-opioid receptor, and so phenomorphan is around 10x more potent than levorphanol, which is itself 6-8x the potency of morphine. Other analogues where the N-(2-phenylethyl) group has been replaced by other aromatic rings. are even more potent, with the N-(2-(2-furyl)ethyl) and the N-(2-(2-thienyl)ethyl) analogues being 60x and 45x stronger than levorphanol, respectively.
==See also==
* 14-Cinnamoyloxycodeinone
* 14-Phenylpropoxymetopon
* 7-PET
* N-Phenethylnormorphine
* N-Phenethylnordesomorphine
* N-Phenethyl-14-ethoxymetopon
* RAM-378
* Ro4-1539
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